发明名称 |
PROCESS FOR THE PREPARATION OF BENZO-USED HETEROARYL SULFAMATES AND CRYSTALLINE FORM OF N-(((2S)-6-CHLORO-2,3-DIHYDRO-L,4-BENZODIOXIN-2-YL) METHYLSULFAMINE |
摘要 |
The present invention is directed to a process for the preparation of benzo-fused heteroaryl sulfamates, useful for the treatment of epilepsy and related disorders according to formula (IA) and to a crystalline compound of formula (I-S). Process for the preparation of a compound of formula (IA). |
申请公布号 |
ZA201007611(B) |
申请公布日期 |
2012.04.25 |
申请号 |
ZA20100007611 |
申请日期 |
2010.10.25 |
申请人 |
JANSSEN PHARMACEUTICA N.V |
发明人 |
ABDEL-MAGID AHMED F;MEHRMAN STEVEN J |
分类号 |
A61K;A61P;C07D |
主分类号 |
A61K |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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