发明名称 |
CARBONATE PRODRUGS AND METHODS OF USING THE SAME |
摘要 |
The present invention provides carbonate prodrugs which comprise a carbonic phosphoric anhydride prodrug moiety attached to the hydroxyl or carboxyl group of a parent drug moiety. The prodrugs may provide improved physicochemical properties over the parent drug. Also provided are methods of treating a disease or condition that is responsive to the parent drug using the carbonate prodrugs, as well as kits and unit dosages. |
申请公布号 |
EP2291084(A4) |
申请公布日期 |
2012.04.25 |
申请号 |
EP20090751525 |
申请日期 |
2009.05.20 |
申请人 |
NEUROGESX, INC. |
发明人 |
MUHAMMAD, NAWEED;BLEY, KEITH, R. |
分类号 |
C07F9/09;A61K31/661;A61P25/02 |
主分类号 |
C07F9/09 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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