发明名称 Sulfonylamino-derivatives as novel inhibitors of histone deacetylase
摘要 This invention comprises the novel compounds of formula (I) wherein n, m, t, R1, R2, R3, R4, R5, L, Q, X, Y, Z and have defined meanings, having histone deacetylase inhibiting enzymatic activity; their preparation, compositions containing them and their use as a medicine.
申请公布号 US8163733(B2) 申请公布日期 2012.04.24
申请号 US20100724273 申请日期 2010.03.15
申请人 VAN EMELEN KRISTOF;BACKX LEO JACOBUS JOZEF;VAN BRANDT SVEN FRANCISCUS ANNA;ANGIBAUD PATRICK RENE;PILATTE ISABELLE NOELLE CONSTANCE;VERDONCK MARC GUSTAAF CELINE;DE WINTER HANS LOUIS JOS;VAN HEUSDEN JIMMY ARNOLD VIVIANE;JANSSEN PHARMACEUTICA N.V. 发明人 VAN EMELEN KRISTOF;BACKX LEO JACOBUS JOZEF;VAN BRANDT SVEN FRANCISCUS ANNA;ANGIBAUD PATRICK RENE;PILATTE ISABELLE NOELLE CONSTANCE;VERDONCK MARC GUSTAAF CELINE;DE WINTER HANS LOUIS JOS;VAN HEUSDEN JIMMY ARNOLD VIVIANE
分类号 A61K31/55;C07D239/42;A61K31/4025;A61K31/4468;A61K31/451;A61K31/4545;A61K31/496;A61K31/506;A61K31/5377;A61K45/00;A61P1/18;A61P5/00;A61P9/00;A61P11/00;A61P13/08;A61P13/10;A61P13/12;A61P15/00;A61P17/00;A61P19/00;A61P25/00;A61P35/00;A61P35/02;A61P43/00;C07D207/14;C07D211/58;C07D401/04;C07D403/04;C07D405/14;C07D409/14 主分类号 A61K31/55
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