发明名称 |
THIAZOLE OR THIADIZALOE DERIVATIVES FOR USE AS SPHINGOSINE 1-PHOSPHATE 1 (S1P1) RECEPTOR AGONISTS |
摘要 |
Thiazole or thiadizaloe derivatives of formula (I) or pharmaceutical salts thereof having pharmacological activity, processes for their preparation, pharmaceutical compositions containing them and their uses in the treatment of various disorders mediated by S1P1 receptor are disclosed. |
申请公布号 |
US2012094979(A1) |
申请公布日期 |
2012.04.19 |
申请号 |
US201013378809 |
申请日期 |
2010.06.17 |
申请人 |
BAILEY JAMES MATTHEW;DEMONT EMMANUEL HUBERT;LIN XICHEN;REN FENG;SMETHURST CHRISTIAN ALAN PAUL;GLAXO WELLCOME HOUSE |
发明人 |
BAILEY JAMES MATTHEW;DEMONT EMMANUEL HUBERT;LIN XICHEN;REN FENG;SMETHURST CHRISTIAN ALAN PAUL |
分类号 |
A61K31/55;A61K31/433;A61K31/4725;A61P1/00;A61P3/10;A61P9/00;A61P9/10;A61P11/06;A61P17/06;A61P19/02;A61P25/00;A61P29/00;A61P31/12;A61P35/00;A61P35/04;A61P37/06;C07D417/10 |
主分类号 |
A61K31/55 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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