发明名称 COMPOUND HAVING HETERO RING SKELETON, AND PROCESS FOR PRODUCING OPTICALLY ACTIVE COMPOUND USING THE AFOREMENTIONED COMPOUND AS ASYMMETRIC CATALYST
摘要 The present invention provides a compound having a heterocyclic skeleton, which is represented by of the formula (I): wherein R1 and R2 are the same or different and each is a lower alkyl group optionally having substituent(s), an aralkyl group optionally having substituent(s) or an aryl group optionally having substituent(s), or R1 and R2 in combination form, together with the nitrogen atom they are bonded to, a heterocycle optionally having substituent(s) (the heterocycle is optionally condensed with an aromatic hydrocarbon ring); ring A is an imidazole ring condensed with an aromatic ring optionally having substituent(s), or a pyrimidin-4-one ring condensed with an aromatic ring optionally having substituent(s); R3 and R4 are the same or different and each is a lower alkyl group optionally having substituent(s), a lower alkenyl group optionally having substituent(s), a lower alkynyl group optionally having substituent(s), an aralkyl group optionally having substituent(s) or an aryl group optionally having substituent(s), or R3 and R4 in combination form, together with the carbon atoms they are respectively bonded to, a homocycle optionally having substituent(s), or a heterocycle optionally having substituent(s) (the homocycle and heterocycle are optionally condensed with an aromatic hydrocarbon ring); and R5 and R6 are the same or different and each is a hydrogen atom or a lower alkyl group optionally having substituent(s), a tautomer thereof or a salt thereof, and which is useful as a catalyst for an asymmetric synthesis.
申请公布号 US2012095227(A1) 申请公布日期 2012.04.19
申请号 US201013259887 申请日期 2010.04.09
申请人 TAKEMOTO YOSHIJI;MURAKAMI KAZUO;SUMITOMO CHEMICAL COMPANY, LIMITED;KYOTO UNIVERSITY 发明人 TAKEMOTO YOSHIJI;MURAKAMI KAZUO
分类号 C07D239/95;C07D235/30 主分类号 C07D239/95
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