发明名称 QUINAZOLINONE-TYPE COMPOUNDS AS CRTH2 ANTAGONISTS
摘要 This application provides for compounds of the formula Formula I or a pharmaceutically acceptable salt thereof, wherein the individual variables are defined herein, as well as processes to prepare these compounds, pharmaceutical compositions comprising the same and their use in treating disease state associated with the CRTH2 receptor.
申请公布号 WO2012051036(A1) 申请公布日期 2012.04.19
申请号 WO2011US55054 申请日期 2011.10.06
申请人 MERCK SHARP & DOHME CORP.;SCHERING CORPORATION;ASLANIAN, ROBERT, G.;BOYCE, CHRISTOPHER, W.;MAZZOLA, ROBERT, D., JR.;MCKITTRICK, BRIAN, A.;MCCORMICK, KEVIN, D.;PALANI, ANANDAN;QIN, JUN;TANG, HAIQUN;XIAO, DONG;YU, YOUNONG;CALDWELL, JOHN, P.;KELLEY, ELIZABETH HELEN;ZHANG, HONGJUN;SILIPHAIVANH, PHIENG;MACCOSS, RACHEL, N.;METHOT, JOEY, L.;GAUUAN, JOLICIA POLIVINA;JIANG, QIN;LEYHANE, ANDREW, J.;BIJU, PURAKKATTLE JOHNY;DONG, LI;HUANG, XIANHAI;SHAO, NING;ZHOU, WEI;DHONDI, PAWAN, K. 发明人 ASLANIAN, ROBERT, G.;BOYCE, CHRISTOPHER, W.;MAZZOLA, ROBERT, D., JR.;MCKITTRICK, BRIAN, A.;MCCORMICK, KEVIN, D.;PALANI, ANANDAN;QIN, JUN;TANG, HAIQUN;XIAO, DONG;YU, YOUNONG;CALDWELL, JOHN, P.;KELLEY, ELIZABETH HELEN;ZHANG, HONGJUN;SILIPHAIVANH, PHIENG;MACCOSS, RACHEL, N.;METHOT, JOEY, L.;GAUUAN, JOLICIA POLIVINA;JIANG, QIN;LEYHANE, ANDREW, J.;BIJU, PURAKKATTLE JOHNY;DONG, LI;HUANG, XIANHAI;SHAO, NING;ZHOU, WEI;DHONDI, PAWAN, K.
分类号 A01N43/54;C07D239/42;C07D401/04 主分类号 A01N43/54
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