发明名称 Azacytidine analogues and uses thereof
摘要 The present invention is directed toward compounds of Formula (I) as follows: wherein, R is H, R5C(O); R1 is where the crossing dashed line illustrates the bond formed joining R1 to the molecule of Formula (I); R2 and R3 are independently OH or H, provided that R2 and R3 are not simultaneously OH; R4 is H or R5C(O), provided that R and R4 are not simultaneously H; and R5 is a C3-C26 alkenyl, or a pharmaceutical salt thereof. Methods of making and using these compounds are also disclosed.
申请公布号 US8158605(B2) 申请公布日期 2012.04.17
申请号 US20080238125 申请日期 2008.09.25
申请人 SILVERMAN LEWIS;HOLLAND JAMES;MOUNT SINAI SCHOOL OF MEDICINE 发明人 SILVERMAN LEWIS;HOLLAND JAMES
分类号 A01N43/04;A61K31/70 主分类号 A01N43/04
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