发明名称 NEW CRYSTALLINE FORMS OF THE SODIUM SALT OF (4- {4- [5- ( 6 - TRIFLUOROMETHYL - PYRIDIN- 3 - YLAMINO ) - PYRIDIN- 2 -YL] -PHENYL} - CYCLOHEXYL) -ACETIC ACID
摘要 The present invention relates to novel crystalline forms of (4-{4-[5-(6-Trifluoromethyl-pyridin-3-ylamino)-pyridin-2-yl]-phenyl}-cyclohexyl)-acetic acid, sodium and their use in the treatment or prevention of a condition or a disorder associated with DGAT1 activity in animals, particularly humans. It also relates processes for making such novel crystalline forms.
申请公布号 CA2813736(A1) 申请公布日期 2012.04.12
申请号 CA20112813736 申请日期 2011.10.05
申请人 NOVARTIS AG 发明人 SUTTON, PAUL ALLEN;GIRGIS, MICHAEL J.;LIANG, JESSICA;PRASHAD, MAHAVIR;VILLHAUER, EDWIN BERNARD
分类号 C07D401/12;A61K31/415;A61P3/04 主分类号 C07D401/12
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