发明名称 |
Carbinol derivatives having cyclic linker |
摘要 |
[Object] To provide a novel LXR&bgr; agonist that is useful as a preventative and/or therapeutic agent for atherosclerosis; arteriosclerosis such as those resulting from diabetes; dyslipidemia; hypercholesterolemia; lipid-related diseases; inflammatory diseases that are caused by inflammatory cytokines; skin diseases such as allergic skin diseases; diabetes; or Alzheimer's disease. [Solving Means] A carbinol compound represented by the following general formula (I) or salt thereof, or their solvate. |
申请公布号 |
US8153634(B2) |
申请公布日期 |
2012.04.10 |
申请号 |
US20090474799 |
申请日期 |
2009.05.29 |
申请人 |
YAMAGUCHI YUKI;KOURA MINORU;KUROBUCHI SAYAKA;MATSUDA TAKAYUKI;OKUDA AYUMU;SUMIDA HISASHI;WATANABE YUICHIRO;ENOMOTO TAKASHI;SHIBUYA KIMIYUKI;KOWA COMPANY, LTD. |
发明人 |
YAMAGUCHI YUKI;KOURA MINORU;KUROBUCHI SAYAKA;MATSUDA TAKAYUKI;OKUDA AYUMU;SUMIDA HISASHI;WATANABE YUICHIRO;ENOMOTO TAKASHI;SHIBUYA KIMIYUKI |
分类号 |
A61K31/4166;A61K31/4178;A61K31/4355;A61K31/4439;A61K31/497;A61K31/501;A61K31/506;C07D233/72;C07D401/02;C07D401/06;C07D403/02;C07D403/06;C07D405/02;C07D405/14;C07D491/048 |
主分类号 |
A61K31/4166 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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