发明名称 |
SULFAMOYL BENZOIC ACID HETEROBICYCLIC DERIVATIVES AS TRPM8 ANTAGONISTS |
摘要 |
<p>The present invention relates to sulfamoyl benzoic acid heterobicyclic derivatives of the formula (I) or a pharmaceutically acceptable salt thereof or a prodrug thereof, processes for their preparation, pharmaceutical compositions containing them and their use in the treatment of various disorders which are mediated via the TRPM8 receptor.</p> |
申请公布号 |
WO2012042915(A1) |
申请公布日期 |
2012.04.05 |
申请号 |
WO2011JP05588 |
申请日期 |
2011.10.03 |
申请人 |
RAQUALIA PHARMA INC.;KAWAMURA, KIYOSHI;SHISHIDO, YUJI;OHMI, MASASHI |
发明人 |
KAWAMURA, KIYOSHI;SHISHIDO, YUJI;OHMI, MASASHI |
分类号 |
C07D401/12;A61K31/443;A61K31/4439;A61K31/444;A61K31/4709;A61P13/00;A61P25/00;A61P29/00;A61P43/00;C07D209/08;C07D215/12;C07D231/56;C07D249/18;C07D307/79;C07D405/04;C07D405/12;C07D405/14;C07D471/04 |
主分类号 |
C07D401/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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