发明名称 NOVEL METHOD OF PREPARING BENZOIMIDAZOLE DERIVATIVES
摘要 This invention relates to a method of preparing a benzoimidazole derivative at high purity and high yield so as to enable the production of the benzoimidazole derivative compound as an antagonist against a vanilloid reactor-1, and particularly to a method of preparing a benzoimidazole derivative at high purity and high yield, wherein the benzoimidazole derivative is synthesized using a novel intermediate, namely, benzaldehyde, and thereby the preparation process is simple so that it can be applied to production.
申请公布号 WO2012044043(A2) 申请公布日期 2012.04.05
申请号 WO2011KR07109 申请日期 2011.09.27
申请人 DAEWOONG PHARMACEUTICAL CO., LTD.;KIM, IN WOO;KIM, JI DUCK;YOON, HONG CHUL;YOON, HEE KYOON;LEE, BYUNG GOO;LEE, JOON HWAN;LIM, YOUNG MOOK;CHOI, SOO JIN 发明人 KIM, IN WOO;KIM, JI DUCK;YOON, HONG CHUL;YOON, HEE KYOON;LEE, BYUNG GOO;LEE, JOON HWAN;LIM, YOUNG MOOK;CHOI, SOO JIN
分类号 C07D401/10;C07D235/18;C07D401/14;C07D471/04 主分类号 C07D401/10
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