发明名称 |
Triazolopyridine 11-beta hydroxysteroid dehydrogenase type I inhibitors |
摘要 |
Novel compounds are provided which are 11-beta-hydroxysteroid dehydrogenase type I inhibitors. 11-beta-hydroxysteroid dehydrogenase type I inhibitors are useful in treating, preventing, or slowing the progression of diseases requiring 11-beta-hydroxysteroid dehydrogenase type I inhibitor therapy. These novel compounds have the structure: or stereoisomers or prodrugs or pharmaceutically acceptable salts thereof wherein W, L, R3, R3a, R3b and R4 are defined herein. |
申请公布号 |
US8148396(B2) |
申请公布日期 |
2012.04.03 |
申请号 |
US20090424674 |
申请日期 |
2009.04.16 |
申请人 |
LI JAMES J.;HAMANN LAWRENCE G.;WANG HAIXIA;RUAN ZHEMING;COOPER CHRISTOPHER B.;LI JUN;ROBL JEFFREY A.;BRISTOL-MYERS SQUIBB COMPANY |
发明人 |
LI JAMES J.;HAMANN LAWRENCE G.;WANG HAIXIA;RUAN ZHEMING;COOPER CHRISTOPHER B.;LI JUN;ROBL JEFFREY A. |
分类号 |
A01N43/42;A61K31/44;C07D513/02 |
主分类号 |
A01N43/42 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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