发明名称 CRYSTALLINE FORMS OF 6- [2- (METHYLCARBAMOYL) PHENYLSULFANYL] -3-E- [2- (PYRIDIN-2-YL) ETHENYL] INDAZOLE SUITABLE FOR THE TREATMENT OF ABNORMAL CELL GROWTH IN MAMMALS
摘要 Disclosed is a crystalline form of 6-[2-(methylcarbamoyl)phenylsulfanyl]-3-E-[2-(pyridin-2-yl)ethenyl]indazole (compound 1 as depicted), wherein said crystalline form is a substantially pure polymorph of Form XLI having a powder X-ray diffraction pattern comprising a peak at diffraction angle 2 Theta as disclosed in the specification. Also disclosed is a pharmaceutical composition comprising the crystalline form XLI of the compound.
申请公布号 NZ580126(A) 申请公布日期 2012.03.30
申请号 NZ20080580126 申请日期 2008.03.25
申请人 PFIZER PRODUCTS INC. 发明人 MCLAUGHLIN, ROBERT, WILLIAM;CAMPETA, ANTHONY, MICHAEL;CHEKAL, BRIAN, PATRICK;SINGER, ROBERT, ALAN
分类号 C07D401/06;A61K31/4439;A61P35/00 主分类号 C07D401/06
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