发明名称 AZABIPHENYLAMINOBENZOIC ACID DERIVATIVES AS DHODH INHIBITORS
摘要 Disclosed are azabiphenylaminobenzoic acid derivatives represented by general formula (I), such as 5-cyclopropyl-2-(2-phenylpyrimidin-5-ylamino)benzoic acid. Also disclosed is the use of the compounds of formula (I) for treating a pathological disease susceptible to amelioration by inhibition of dihydrooorotate dehydrogenase.
申请公布号 NZ582709(A) 申请公布日期 2012.03.30
申请号 NZ20080582709 申请日期 2008.08.08
申请人 ALMIRALL, S.A. 发明人 CASTRO PALOMINO LARIA, JULIO, CESAR;TERRICABRAS BELART, EMMA;ERRA SOLA, MONTSERRAT;NAVARRO ROMERO, ELOISA;FONQUERNA POU, SILVIA;CARDUS FIGUERAS, ARANZAZU;LOZOYA TORIBIO, MARIA, ESTRELLA
分类号 A61P31/00;A61K31/44;A61K31/506;A61P17/00;A61P19/00;A61P35/00;A61P37/00;C07D213/74;C07D239/42;C07D401/04;C07D401/10;C07D413/10 主分类号 A61P31/00
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