发明名称 CYCLIC-ALKYLAMINE DERIVATIVES AS INHIBITORS OF THE INTERACTION BETWEEN MDM2 AND P53
摘要 The present invention provides compounds of formula (I), their use as an inhibitor of a p53-MDM2 interaction as well as pharmaceutical compositions comprising said compounds of formula (I) wherein n, m, p, t, R1, R2, R3, R4, R5, R6, R7, Q, Y and Z have defined meanings.
申请公布号 US2012071508(A1) 申请公布日期 2012.03.22
申请号 US201113307153 申请日期 2011.11.30
申请人 LACRAMPE JEAN FERNAND ARMAND;MEYER CHRISTOPHE;SCHOENTJES BRUNO;PONCELET ALAIN PHILIPPE;WERMUTH CAMILLE GEORGES;GIETHLEN BRUNO;CONTRERAS JEAN-MARIE;JOUBERT MURIEL;VAN HIJFTE LUC 发明人 LACRAMPE JEAN FERNAND ARMAND;MEYER CHRISTOPHE;SCHOENTJES BRUNO;PONCELET ALAIN PHILIPPE;WERMUTH CAMILLE GEORGES;GIETHLEN BRUNO;CONTRERAS JEAN-MARIE;JOUBERT MURIEL;VAN HIJFTE LUC
分类号 A61K31/4709;A61K31/435;A61K31/4439;A61P35/00;C07D401/14 主分类号 A61K31/4709
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