发明名称 |
CONDENSED HETEROCYCLIC DERIVATIVE HAVING MELANINE-CONCENTRATING HORMONE RECEPTOR ANTAGONISTIC ACTIVITY |
摘要 |
<p>Provided is a novel compound which has MCH R1 receptor antagonistic activity and is represented by formula (I), a pharmaceutically acceptable salt thereof, or a solvate of the same. (In the formula, the portion AA represented by formula (1) is BB etc., the broken lines indicate whether or not a bond is present, X1 is O or S, when the broken lines joined to X2 indicate that a bond is not present, X2 is N or C(R3), X4-X3-X2 is X4-O-C(R4)(R4)-C(R4)(R4)-X2 etc., -Y1- is a single bond etc., -Y2- is a single bond etc., each R2 is independently a halogen etc., R3 is hydrogen etc., R4 is hydrogen etc., D is an alkyl etc., ring B is a cycloalkyl etc., p is an integer of 0 to 4, and q is an integer of 1 to 4.</p> |
申请公布号 |
WO2012036233(A1) |
申请公布日期 |
2012.03.22 |
申请号 |
WO2011JP71093 |
申请日期 |
2011.09.15 |
申请人 |
SHIONOGI & CO., LTD.;OMORI, NAOKI;OHDAN, MASAHIDE;WADA, TOSHIHIRO;KATO, TERUKAZU;TANAKA, NOBUYUKI;YOSHIDA, YUTAKA;SATO, HIROKI;MURASHI, TAKAMI |
发明人 |
OMORI, NAOKI;OHDAN, MASAHIDE;WADA, TOSHIHIRO;KATO, TERUKAZU;TANAKA, NOBUYUKI;YOSHIDA, YUTAKA;SATO, HIROKI;MURASHI, TAKAMI |
分类号 |
C07D223/16;A61K31/4025;A61K31/517;A61K31/536;A61K31/5365;A61K31/5377;A61K31/538;A61K31/5383;A61K31/55;A61K31/553;A61P3/04;A61P3/10;A61P5/00;A61P9/10;A61P15/10;A61P19/02;A61P25/28;A61P43/00;C07D239/96;C07D265/22;C07D265/36;C07D267/14;C07D311/36;C07D413/04;C07D413/12;C07D413/14;C07D471/04;C07D498/04;C07D513/04 |
主分类号 |
C07D223/16 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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