发明名称 |
3-AZA-6,8-DIOXABICYCLO[3.2.1]OCTANES AND ANALOGUES AND COMBINATORIAL LIBRARIES |
摘要 |
The present invention relates to new highly functionalized heterobicycle derivatives of general formula (I), prepared by a process which involves only two steps by using, as starting products, commercially available, or easily prepared, .alpha.-amino ketones and .alpha.,.beta.-dihydroxy acids or .alpha.-amino-.beta.-hydroxy acids or .alpha.-hydroxy-.beta.-amino acids or .alpha.,.beta.-dithiol acids derivatives and to libraries containing compounds of formula (I) and to the generation of such combinatorial libraries composed of compounds of formula (I), in individual synthesis, mixture synthesis, split and recombine synthesis and parallel synthesis either in manual or automated fashion.
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申请公布号 |
CA2401693(C) |
申请公布日期 |
2012.03.20 |
申请号 |
CA20012401693 |
申请日期 |
2001.02.27 |
申请人 |
UNIVERSITA' DEGLI STUDI DI FIRENZE |
发明人 |
GUARNA, ANTONIO;MENCHI, GLORIA;OCCHIATO, ERNESTO GIOVANNI;MACHETTI, FABRIZIO;SCARPI, DINA |
分类号 |
C07D498/08;C07D241/00;C07D263/00;C07D265/00;C07D317/00;C07D513/08 |
主分类号 |
C07D498/08 |
代理机构 |
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