发明名称 |
PRODUCTION METHOD OF PHENACYL BROMIDE DERIVATIVE |
摘要 |
<P>PROBLEM TO BE SOLVED: To provide an induction production method of a phenacyl bromide derivative (II) useful as a synthetic intermediate body of a 2-isoindole derivative which is an excellent thrombin receptor antagonistic agent. <P>SOLUTION: The production method of a compound expressed by a formula (II) includes a process for obtaining the compound expressed by the formula (II) by reacting a compound expressed by a formula (I) with a tribromide compound. <P>COPYRIGHT: (C)2012,JPO&INPIT |
申请公布号 |
JP2012051866(A) |
申请公布日期 |
2012.03.15 |
申请号 |
JP20100198110 |
申请日期 |
2010.09.03 |
申请人 |
EISAI R & D MANAGEMENT CO LTD |
发明人 |
YAMAZAKI SHIGEYA;MARUO MASAFUMI;HOSOYA TAKESHI;YOSHIKAWA TAICHI;AKIYAMA TOSHIHIKO;KAYANO AKIO |
分类号 |
C07D295/10 |
主分类号 |
C07D295/10 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|