<p>Disclosed are 4-amino-2-butenamides of Formula (I) having pharmacological activity, pharmaceutical compositions containing them, and methods for the treatment of diseases mediated by the cathepsin C enzyme such as chronic obstructive pulmonary disease.</p>
申请公布号
MX2012001797(A)
申请公布日期
2012.03.14
申请号
MX20120001797
申请日期
2010.08.11
申请人
GLAXO GROUP LIMITED.*
发明人
BUSCH-PETERSEN, JAKOB;PALOVICH, MICHAEL R.;NEVINS, NEYSA;LI, HUIJIE;ANDERSON, NIALL;EVANS, BRIAN;SOLLIS, STEVEN L.;WALL, MICHAEL D.;BULLION, ANN M.