发明名称 |
NOVEL CRYSTALLINE HYDRATE, AMORPHOUS AND POLYMORPHIC FORMS OF DIHYDRO-BENZOXAZOLE-6-YL-ACETAMIDE DERIVATIVE AND PROCESSES FOR THEIR PREPARATION |
摘要 |
The invention relates to novel crystalline hydrate, amorphous and crystalline polymorphic forms of 2-[4-(4-Fluoro-benzyl)-piperidine-1-yl]-2-oxo-N-(2-oxo-2,3-dihydro-benzoxazole-6-yl)-acetamide (I) (radiprodil). Processes for the preparation of these forms, compositions containing these forms, and methods of use thereof are also described. |
申请公布号 |
US2012059034(A1) |
申请公布日期 |
2012.03.08 |
申请号 |
US201013147181 |
申请日期 |
2010.03.01 |
申请人 |
DEMETER ADAM;NEMET ZOLTAN;NEMES ANDRAS;SEBOK FERENC;BARTANE SZALAI GIZELLA;CZIBULA LASZLO |
发明人 |
DEMETER ADAM;NEMET ZOLTAN;NEMES ANDRAS;SEBOK FERENC;BARTANE SZALAI GIZELLA;CZIBULA LASZLO |
分类号 |
A61K31/454;A61P11/00;A61P11/06;A61P25/00;A61P25/04;A61P25/08;A61P25/16;A61P25/22;A61P25/24;A61P25/28;A61P25/32;A61P25/36;A61P27/06;A61P27/16;C07D413/12 |
主分类号 |
A61K31/454 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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