发明名称 |
BENZOIC ACID, BENZOIC ACID DERIVATIVES AND HETEROARYL CARBOXYLIC ACID CONJUGATES OF HYDROCODONE, PRODRUGS, METHODS OF MAKING AND USE THEREOF |
摘要 |
The presently described technology provides compositions comprising aryl carboxylic acids chemically conjugated to hydrocodone (morphinan-6-one, 4,5-alpha-epoxy-3-methoxy-17-methyl) to form novel prodrugs/compositions of hydrocodone, including benzoates and heteroaryl carboxylic acids, which have a decreased potential for abuse of hydrocodone. The present technology also provides methods of treating patients, pharmaceutical kits and methods of synthesizing conjugates of the present technology. |
申请公布号 |
SG177445(A1) |
申请公布日期 |
2012.02.28 |
申请号 |
SG20110097482 |
申请日期 |
2010.07.01 |
申请人 |
KEMPHARM, INC. |
发明人 |
MICKLE, TRAVIS;GUENTHER, SVEN;MICKLE, CHRISTAL;CHI, GUOCHEN;KANSKI, JAROSLAW;MARTIN, ANDREA K.;BERA, BINDU |
分类号 |
|
主分类号 |
|
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|