发明名称 PREPARATION OF 3-AMINO-3-(CYCLOBUTYLMETHYL)-2-(HYDROXY)-PROPIONAMIDE HYDROCHLORIDE
摘要 <p>AbstractPREPARATION OF 3-AMINO-3-(CYCLOBUTYLMETHYL)-2-(HYDROXY)- PROPIONAMIDE HYDROCHLORIDEDisclosed is a process for preparing 3-(amino)-3-cyclobutylmethyl-2-hydroxy-propionamide hydrochlo ride, an intermediate useful in the preparation of the HCV protease inhibitor (1R,5S)-N-[3-amino-1-(cyclobutyl-methyl)-2,3-dioxopropyl]-3-[2(S)-[[[(1,1-dimethylethyl)aminoIcarbonyl]amino]-3,3-dimethyl-1-oxobutyl]-6,6-dimethyl-3-azabi-cyclo[3.1.0]hexan-2(S)-carboxamide.No Figure.</p>
申请公布号 SG177906(A1) 申请公布日期 2012.02.28
申请号 SG20110094364 申请日期 2007.12.17
申请人 SCHERING CORPORATION (US) 发明人 PARK, JEONGHAN;VATER, EUGENE, J.;DONG, SHUAN;IWAMA, TETSUO;RAGHAVAN, RAMANI, R.;LEE, HONG-CHANG;WONG, GEORGE, S. K.
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