摘要 |
具式(I)之化合物:X-Ser-Asp-Ala-Ala-Val-Asp-Thr-Ser-(I)Ser-Glu-Ile-Thr-Thr-Lys-Asp-Leu-Z其中该X为乙醯基或焦麸胺醯基而Z为-NH2、-Lys- Glu-Lys-Lys-Glu-Val-Val-Glu-Clu-Ala-Glu-Asn-Pro- NH2、-Lys-Glu-Lys-Lys-Glu-Val-Val-Glu-Glu-Ala-Glu-Asn-Gly-NH2或-Lys-Glu-Lys-Lys-Glu-Val-Val-Glu- G1u-Ala-Glu-Asn其限制条件为,当X为焦麸胺醯基时,;而且当X为乙醯基时,Z便非-Lys-Glu-Lys-Lys- Glu-Val-Val-Glu-Glu~Ala-G1u-Asn及其制法。 |