发明名称 |
PROCESS FOR SUBSTITUTED 3-AMINO-5-OXO-4,5-DIHYDRO-[1,2,4]TRIAZINE S. |
摘要 |
<p>Processes including preparation of trans-4-[(3-amino-5-oxo-4,5-dihydro-[1,2,4]triazin-6-ylm ethyl)-carbamoyl]-cyclohexanecarboxylic acid methyl ester, and its conversion to trans-4-(4-amino-5-susbtituted-imidazo[5,1-Æ ][1,2,4]tri azin-7-yl)-cyclohexanecarboxylic acid compounds.</p> |
申请公布号 |
MX2012000431(A) |
申请公布日期 |
2012.02.21 |
申请号 |
MX20120000431 |
申请日期 |
2010.07.08 |
申请人 |
OSI PHARMACEUTICALS, LLC |
发明人 |
DONG, HANQING;MULVIHILL, KRISTEN MICHELLE;WERNER, DOUGLAS S.;RECHKA, JOSEF A.;MAO, YUNYU |
分类号 |
C07D253/06;C07D403/04;C07D487/04 |
主分类号 |
C07D253/06 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|