发明名称 ACID ADDITION SALTS OF THE 2-[2-[[(4-METHOXY-2,6-DIMETHYLPHENYL)SULFONYL]-(METHYL)AMINO]ETHOXY]-N-METHYL-N-[3-(4-METHYLPIPERAZIN-1-YL)CYCLOHEXYL] ACETAMIDE AND THE USE THEREOF AS BRADYKININ B1 RECEPTOR ANTAGONISTS
摘要 The invention relates to the novel acid addition salts AB of the following free base of formula (A) or the enantiomer thereof with a physiologically acceptable acid B selected from the group consisting of hydrochloric acid, fumaric acid, and tartaric acid and to the polymorphs, hydrates, and solvates thereof.
申请公布号 WO2012017027(A1) 申请公布日期 2012.02.09
申请号 WO2011EP63413 申请日期 2011.08.04
申请人 BOEHRINGER INGELHEIM INTERNATIONAL GMBH;PACHUR, THORSTEN;PFRENGLE, WALDEMAR;BIRK, MANFRED;SCHNAUBELT, JUERGEN;WERTHMANN, ULRIKE 发明人 PACHUR, THORSTEN;PFRENGLE, WALDEMAR;BIRK, MANFRED;SCHNAUBELT, JUERGEN;WERTHMANN, ULRIKE
分类号 C07D295/135;A61K31/495;A61P29/00 主分类号 C07D295/135
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