发明名称 CRYSTALLINE AND AMORPHOUS FORMS OF ALMOREXANT HYDROCHLORIDE AND A METHOD OF THEIR PREPARATION
摘要 The invention relates to crystalline and amorphous forms of (2R)-2-{(1S)-6,7-dimethoxy-1-[2-(4-trifluoromethyl-phenyl)-ethyl] -3,4-dihydro- 1H-isoquinolin-2-yl} -N-methyl-2-phenyl- acetamide hydrochloride (I) (almorexant) and a method of their preparation.
申请公布号 WO2011063773(A3) 申请公布日期 2012.02.02
申请号 WO2010CZ00119 申请日期 2010.11.24
申请人 ZENTIVA, K.S.;RADL, STANISLAV;CERNY, JOSEF;BRUSOVA, HANA 发明人 RADL, STANISLAV;CERNY, JOSEF;BRUSOVA, HANA
分类号 C07D217/18;A61K31/472;A61P25/20 主分类号 C07D217/18
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