CRYSTALLINE AND AMORPHOUS FORMS OF ALMOREXANT HYDROCHLORIDE AND A METHOD OF THEIR PREPARATION
摘要
The invention relates to crystalline and amorphous forms of (2R)-2-{(1S)-6,7-dimethoxy-1-[2-(4-trifluoromethyl-phenyl)-ethyl] -3,4-dihydro- 1H-isoquinolin-2-yl} -N-methyl-2-phenyl- acetamide hydrochloride (I) (almorexant) and a method of their preparation.
申请公布号
WO2011063773(A3)
申请公布日期
2012.02.02
申请号
WO2010CZ00119
申请日期
2010.11.24
申请人
ZENTIVA, K.S.;RADL, STANISLAV;CERNY, JOSEF;BRUSOVA, HANA