发明名称 |
Process for the preparation of (2R,3S)-3-phenylisoserine methyl ester acetate salt |
摘要 |
A process for the enantioselective preparation of (2R,3S)-3-phenylisoserine methyl ester acetate salt of formula (I) which is an useful building block for the synthesis of taxane derivatives. The process involves the resolution of racemic threo-phenylisoserine amide and its conversion into (I). |
申请公布号 |
US8106231(B2) |
申请公布日期 |
2012.01.31 |
申请号 |
US20080527887 |
申请日期 |
2008.02.11 |
申请人 |
CICERI DANIELE;GABETTA BRUNO;VIGNOLA NICOLA;MITZEL FRIEDER;WEBER BEAT T.;INDENA S.P.A. |
发明人 |
CICERI DANIELE;GABETTA BRUNO;VIGNOLA NICOLA;MITZEL FRIEDER;WEBER BEAT T. |
分类号 |
C07C229/00 |
主分类号 |
C07C229/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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