发明名称 |
Bisamide inhibitors of hedgehog signaling |
摘要 |
The invention provides inhibitors of hedgehog signaling that are useful as a therapeutic agents for treating malignancies where the compounds have the general formula I: wherein ring A, ring B, R1, R2, R3, R4, R5, m and n are as defined herein. |
申请公布号 |
US8101610(B2) |
申请公布日期 |
2012.01.24 |
申请号 |
US20060093530 |
申请日期 |
2006.11.14 |
申请人 |
GOLDSMITH RICHARD A.;SUTHERLIN DANIEL P.;ROBARGE KIRK D.;OLIVERO ALAN G.;GENENTECH, INC.;CURIS INC. |
发明人 |
GOLDSMITH RICHARD A.;SUTHERLIN DANIEL P.;ROBARGE KIRK D.;OLIVERO ALAN G. |
分类号 |
A61K31/505;A61K31/4164;A61K31/4196;A61K31/4965;C07D213/81 |
主分类号 |
A61K31/505 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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