METHOD FOR PREPARING SITAGLIPTIN AND AMINE SALT INTERMEDIATES USED THEREIN
摘要
The present invention relates to a method for preparing sitagliptin by using an amine salt of (3R)-3-azido-4-(2,4,5-trifluorophenyl)-butyric acid (formula (V)) in a high yield and purity, and amine salt intermediates used therein.
申请公布号
WO2011102640(A3)
申请公布日期
2012.01.19
申请号
WO2011KR01024
申请日期
2011.02.16
申请人
HANMI HOLDINGS CO., LTD.;CHANG, JI-YEON;LEE, HYUN SEUNG;KIM, DONG JUN;KO, MYOUNG-SIL;KIM, NAM DU;CHANG, YOUNG KIL;KIM, MAENG SUP
发明人
CHANG, JI-YEON;LEE, HYUN SEUNG;KIM, DONG JUN;KO, MYOUNG-SIL;KIM, NAM DU;CHANG, YOUNG KIL;KIM, MAENG SUP