发明名称 |
Crystallisation process for 1-(beta-D-glucopyranosyl)-4-methyl-3- [5-(4-fluorophenyl)-2-thienylmethyl] benzene |
摘要 |
The present invention relates to a crystallisation procedure to obtain 1 -(β-D-glucopyranosyl)-4-methyl-3-[5-(4-fluorophenyl)-2-thienylmethyl] benzene hemihydrate crystals having a narrow particle size distribution and improved flowability, bulk and tap density properties. |
申请公布号 |
AU2010270202(A1) |
申请公布日期 |
2012.01.19 |
申请号 |
AU20100270202 |
申请日期 |
2010.07.08 |
申请人 |
JANSSEN PHARMACEUTICA NV |
发明人 |
RAMMELOO, THOMAS JOACHIM LANDEWALD;DE KEYSER, RUBEN;SCHILDERMANS, GUSTAAF JOZEF PETRUS |
分类号 |
C07D309/10 |
主分类号 |
C07D309/10 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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