发明名称 SOLID DISPERSION OF ALFA-KETOAMIDE DERIVATIVES
摘要 A solid dispersion comprising ((1S)-1-((((1S)-1-benzyl-2,3-dioxo-3-(cyclopropylamino)propyl)amino)carbonyl)-3-methylbutyl)carbamic acid 5-methoxy-3-oxapentyl ester made amorphous in the presence of a water-soluble cellulosic polymer has improved storage stability. The solid dispersion also has improved solubility for an improved bioavailability.
申请公布号 WO2012008159(A1) 申请公布日期 2012.01.19
申请号 WO2011JP04021 申请日期 2011.07.13
申请人 SENJU PHARMACEUTICAL CO., LTD.;CHEN, XIAN ANDREW;FAN, JOHN;YAMAGUCHI, MASAZUMI 发明人 CHEN, XIAN ANDREW;FAN, JOHN;YAMAGUCHI, MASAZUMI
分类号 A61K9/19;A61K31/165;A61K47/38 主分类号 A61K9/19
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