发明名称 PYRAZOLO [1, 5A] PYRIMIDINE AND THIENO [3, 2B] PYRIMIDINE DERIVATIVES AS IRAK4 MODULATORS
摘要 Compounds of the formula I or II: wherein X, m, Ar, R1 and R2 are as defined herein. The subject compounds are useful for treatment of IRAK-mediated conditions.
申请公布号 CA2802641(A1) 申请公布日期 2012.01.19
申请号 CA20112802641 申请日期 2011.07.08
申请人 F. HOFFMANN-LA ROCHE AG 发明人 ARORA, NIDHI;CHEN, SHAOQING;HERMANN, JOHANNES CORNELIUS;KUGLSTATTER, ANDREAS;LABADIE, SHARADA SHENVI;LIN, CLARA JEOU JEN;LUCAS, MATTHEW C.;MOORE, AMY GERALDINE;PAPP, EVA;TALAMAS, FRANCISCO XAVIER;WANNER, JUTTA;ZHAI, YANSHENG
分类号 C07D487/04;A61K31/4365;A61K31/519;A61P11/00;A61P29/00;C07D495/04 主分类号 C07D487/04
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