发明名称 Chemical Compounds
摘要 The invention relates to sulfonamide derivatives, to their use in medicine, to compositions containing them, to processes for their preparation and to intermediates used in such processes. More particularly the invention relates to a new sulfonamide Nav1.7 inhibitors of formula (I): or a pharmaceutically acceptable salt thereof, wherein Het1, X, R1, R2, R3, R4 and R5 are as defined in the description. Nav 1.7 inhibitors are potentially useful in the treatment of a wide range of disorders, particularly pain.
申请公布号 US2012010183(A1) 申请公布日期 2012.01.12
申请号 US201113179587 申请日期 2011.07.11
申请人 BELL ANDREW SIMON;BROWN ALAN DANIEL;DE GROOT MARCEL JOHN;LEWTHWAITE RUSSELL ANDREW;MARSH IAN ROGER;MILLAN DAVID SIMON;PACHECO MANUEL PEREZ;RAWSON DAVID JAMES;SCIAMMETTA NUNZIO;STORER ROBERT IAN;SWAIN NIGEL ALAN;GAULIER STEVEN MATTHIEU;PFIZER LIMITED 发明人 BELL ANDREW SIMON;BROWN ALAN DANIEL;DE GROOT MARCEL JOHN;LEWTHWAITE RUSSELL ANDREW;MARSH IAN ROGER;MILLAN DAVID SIMON;PACHECO MANUEL PEREZ;RAWSON DAVID JAMES;SCIAMMETTA NUNZIO;STORER ROBERT IAN;SWAIN NIGEL ALAN;GAULIER STEVEN MATTHIEU
分类号 A61K31/44;A61K31/416;A61K31/4427;A61K31/4439;A61K31/4545;A61K31/47;A61K31/506;A61P29/00;C07D213/69;C07D215/20;C07D231/56;C07D401/04;C07D401/12;C07D405/12 主分类号 A61K31/44
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