发明名称 SOLID STATE FORMS OF ETORICOXIB SALTS
摘要 <p>Provided herein are novel solid state forms of etoricoxib salts, process for their preparation, pharmaceutical compositions, and method of treating thereof. The etoricoxib salts include an oxalate salt, a succinate salt, a fumarate salt, a besylate salt, a hydrobromide salt, a glutamate salt, a sulfamate salt, a benzoate salt, a cinnamate salt, a salicylate salt, or a tosylate salt. The solid state forms of etoricoxib salts disclosed herein are useful for preparing etoricoxib free base with high purity.</p>
申请公布号 WO2012004677(A1) 申请公布日期 2012.01.12
申请号 WO2011IB02278 申请日期 2011.07.05
申请人 ACTAVIS GROUP PTC EHF;KHUNT, MAYUR, DEVJIBHAI;SUBBARAO, ATHUKURI, VENKATA;PRADHAN, NITIN, SHARADCHANDRA;VARMA, SHRIKANT, MURLIDHAR 发明人 KHUNT, MAYUR, DEVJIBHAI;SUBBARAO, ATHUKURI, VENKATA;PRADHAN, NITIN, SHARADCHANDRA;VARMA, SHRIKANT, MURLIDHAR
分类号 C07D213/61;A61K31/444;A61P29/00 主分类号 C07D213/61
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