发明名称 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT
摘要 <p>Compounds having activity as phosphate transport inhibitors, more specifically, inhibitors of intestinal apical membrane Na/phosphate co-transport, are disclosed. The compounds have the following structure (I): including stereoisomers, pharmaceutically acceptable salts and prodrugs thereof, wherein X, Y and A are as defined herein. Methods associated with preparation and use of such compounds, as well as pharmaceutical compositions comprising such compounds, are also disclosed.</p>
申请公布号 WO2012006474(A2) 申请公布日期 2012.01.12
申请号 WO2011US43262 申请日期 2011.07.07
申请人 ARDELYX, INC.;LEWIS, JASON, G.;JACOBS, JEFFREY, W.;REICH, NICHOLAS;LEADBETTER, MICHAEL, R.;BELL, NOAH;CHANG, HAN-TING;CHEN, TAO;NAVRE, MARC;CHARMOT, DOMINIQUE;CARRERAS, CHRISTOPHER;LABONTE, ERIC 发明人 LEWIS, JASON, G.;JACOBS, JEFFREY, W.;REICH, NICHOLAS;LEADBETTER, MICHAEL, R.;BELL, NOAH;CHANG, HAN-TING;CHEN, TAO;NAVRE, MARC;CHARMOT, DOMINIQUE;CARRERAS, CHRISTOPHER;LABONTE, ERIC
分类号 C07D403/02 主分类号 C07D403/02
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