发明名称 THERAPEUTIC USES OF DERIVATIVES OF PIPERIDINYL-AND PIPERIDINYL-ALKYL CARBAMATES
摘要 Compound corresponding to the general formula (I): in which A=N or CR2; R2═H, F, OH, CN, CF3, C1-6-alkyl, C1-6-alkoxy; n=2 or 3 and m=2 when A=N; n=1, 2 or 3 and m=1 or 2 when A=CR2; B=covalent bond or C1-8-alkylene; R1=optionally substituted heteroaryl; R3═CHR4CONHR5; R4═H or C1-6-alkyl; R5═H, C1-6-alkyl, C3-7-cycloalkyl, C3-7-cycloalkyl-C1-C6-alkylene; in the form of a base, an acid-addition salt, a hydrate or a solvate. Therapeutic uses thereof.
申请公布号 US2012004207(A1) 申请公布日期 2012.01.05
申请号 US201113229106 申请日期 2011.09.09
申请人 ABOUABDELLAH AHMED;BURNIER PHILIPPE;HOORNAERT CHRISTIAN;JEUNESSE JEAN;PUECH FREDERIC;SANOFI-AVENTIS 发明人 ABOUABDELLAH AHMED;BURNIER PHILIPPE;HOORNAERT CHRISTIAN;JEUNESSE JEAN;PUECH FREDERIC
分类号 A61K31/495;A61K31/397;A61K31/435;A61K31/436;A61K31/44;A61K31/496;A61K31/497;A61K31/501;A61K31/506;A61K31/551;A61P1/00;A61P1/08;A61P3/00;A61P9/00;A61P9/10;A61P13/00;A61P19/10;A61P25/00;A61P25/08;A61P25/28;A61P27/02;A61P29/00;A61P31/00;A61P31/04;A61P31/12;A61P33/00;A61P35/00;A61P37/00;A61P37/08;C07D211/26;C07D213/38;C07D295/12;C07D295/13;C07D295/15;C07D401/04;C07D401/12;C07D401/14;C07D403/12;C07D403/14;C07D413/04;C07D417/04;C07D417/12;C07D471/04;C07D491/04;C07D491/048;C07D495/04 主分类号 A61K31/495
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