发明名称 |
FUNCTIONALLY SELECTIVE LIGANDS OF DOPAMINE D2 RECEPTORS |
摘要 |
The present invention relates to novel functionally selective ligands of dopamine D2 receptors, including agonists, antagonists, and inverse agonists. The invention further relates to the use of these compounds for treating central nervous system disorders related to D2 receptors. |
申请公布号 |
WO2012003418(A2) |
申请公布日期 |
2012.01.05 |
申请号 |
WO2011US42734 |
申请日期 |
2011.07.01 |
申请人 |
THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL;JIN, JIAN;ROTH, BRYAN;FRYE, STEPHEN |
发明人 |
JIN, JIAN;ROTH, BRYAN;FRYE, STEPHEN |
分类号 |
C07D401/12;A61K31/4375;A61K31/4709;A61P25/00;C07D417/12;C07D471/04 |
主分类号 |
C07D401/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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