发明名称 NEW BENZOTHIAZINONE DERIVATIVES AND THEIR USE AS ANTIBACTERIAL AGENTS
摘要 Novel benzothiazin derivatives of formula (I) and their use as antibacterial agents in infectious diseases caused by bacteria, especially tuberculosis (TB) and leprosy caused by mycobacteria, wherein Rand Rare, independently each from other, NO, CN, trifluoromethyl, halogen, CONRR, COOR, CHO, SONRR, or OCF; Rand Rare, independently each from other, H or a methyl group; Rand Rare, independently each from other, linear or branched aliphatic radical having 1-8 chain members, or Rand Rtogether represent a bivalent radical -(CR)wherein m is 1-4, or Rand Rtogether represent a bivalent radical defined in the invention claims; R, Rand Rare, independently each from other, H or a linear or branched aliphatic radical having 1-7 chain members or phenyl.
申请公布号 EA015910(B1) 申请公布日期 2011.12.30
申请号 EA20080070564 申请日期 2006.05.24
申请人 LEIBNIZ INSTITUTE FOR NATURAL PRODUCT RESEARCH AND INJECTION BIOLOGY E.V.HANS-KNOLL-INSTITUT (HKI) 发明人 MAKAROV VADIM, A.;COLE ETEWART, T.;MOLLMANN UTE
分类号 C07D417/04;A61K31/5415;A61P31/04;C07D491/10 主分类号 C07D417/04
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