发明名称 |
2-[5-BROMO-4-CYCLOPROPYL NAPHTHALEN-1-YL)-4H-[1, 2, 4]TRIAZOL-3-YLSULFANYL] ACETIC ACID METHYL ESTER |
摘要 |
There presented 2-[5-Bromo-4-(4-cyclopropylnaphthalen-1-yl)-4H-[1,2,4]triazol-3-ylsulfanyl]acetic acid methyl ester for preparing S-triazolyl-α-mercaptoacetanilides as inhibitors of HIV reverse transcriptase and are useful in the treatment of HIV infections. |
申请公布号 |
EA015846(B1) |
申请公布日期 |
2011.12.30 |
申请号 |
EA20090001186 |
申请日期 |
2005.08.25 |
申请人 |
ARDEA BIOSCIENCES, INC. |
发明人 |
GIRARDET JEAN-LUC;KOH YUNG-HYO;DE LA ROSE MARTHA;GUNIC ESMIR;HONG ZHI;LANG STANLEY;KIM HONG, WOO |
分类号 |
C07D249/12;A61K31/4196;A61P31/18;C07D249/14 |
主分类号 |
C07D249/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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