发明名称 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY
摘要 The present invention relates to substituted triazole compounds and compositions comprising substituted triazole compounds. The invention further relates to methods of inhibiting the activity of Hsp90 in a subject in need thereof and methods for preventing or treating hyperproliferative disorders, such as cancer, in a subject in need thereof comprising administering to the subject a substituted triazole compound of the invention, or a composition comprising such a compound.
申请公布号 US2011319447(A1) 申请公布日期 2011.12.29
申请号 US201113229178 申请日期 2011.09.09
申请人 SUN LIJUN;YING WEIWEN;CHAE JUNGHYUN;PRZEWLOKA TERESA;ZHANG SHIJIE;CHIMMANAMADA DINESH U.;FOLEY KEVIN;DU ZHENJIAN;LI HAO;JAMES DAVID;NG HOWARD P.;DEMKO ZACHARY;ZHOU DAN;QIN SHUZHEN;SYNTA PHARMACEUTICALS CORP. 发明人 SUN LIJUN;YING WEIWEN;CHAE JUNGHYUN;PRZEWLOKA TERESA;ZHANG SHIJIE;CHIMMANAMADA DINESH U.;FOLEY KEVIN;DU ZHENJIAN;LI HAO;JAMES DAVID;NG HOWARD P.;DEMKO ZACHARY;ZHOU DAN;QIN SHUZHEN
分类号 A61K31/4709;A61K31/4196;A61K31/422;A61P35/00;C07D403/12;C07D403/14;C07D413/14 主分类号 A61K31/4709
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