发明名称 |
TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY |
摘要 |
The present invention relates to substituted triazole compounds and compositions comprising substituted triazole compounds. The invention further relates to methods of inhibiting the activity of Hsp90 in a subject in need thereof and methods for preventing or treating hyperproliferative disorders, such as cancer, in a subject in need thereof comprising administering to the subject a substituted triazole compound of the invention, or a composition comprising such a compound.
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申请公布号 |
US2011319447(A1) |
申请公布日期 |
2011.12.29 |
申请号 |
US201113229178 |
申请日期 |
2011.09.09 |
申请人 |
SUN LIJUN;YING WEIWEN;CHAE JUNGHYUN;PRZEWLOKA TERESA;ZHANG SHIJIE;CHIMMANAMADA DINESH U.;FOLEY KEVIN;DU ZHENJIAN;LI HAO;JAMES DAVID;NG HOWARD P.;DEMKO ZACHARY;ZHOU DAN;QIN SHUZHEN;SYNTA PHARMACEUTICALS CORP. |
发明人 |
SUN LIJUN;YING WEIWEN;CHAE JUNGHYUN;PRZEWLOKA TERESA;ZHANG SHIJIE;CHIMMANAMADA DINESH U.;FOLEY KEVIN;DU ZHENJIAN;LI HAO;JAMES DAVID;NG HOWARD P.;DEMKO ZACHARY;ZHOU DAN;QIN SHUZHEN |
分类号 |
A61K31/4709;A61K31/4196;A61K31/422;A61P35/00;C07D403/12;C07D403/14;C07D413/14 |
主分类号 |
A61K31/4709 |
代理机构 |
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地址 |
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