发明名称 |
PROCESSES AND INTERMEDIATES FOR THE PREPARATION OF ASPARTIC ACETAL CASPASE INHIBITORS |
摘要 |
<p>The invention relates to
a process of producing a compound of
comprising purifying a mixture of
wherein R 8 is a protecting group, and purifying includes chromatographing, selectively crystallizing, or dynamically crystallizing the mixture.</p> |
申请公布号 |
KR20110137409(A) |
申请公布日期 |
2011.12.22 |
申请号 |
KR20117029981 |
申请日期 |
2005.03.11 |
申请人 |
VERTEX PHARMACEUTICALS INCORPORATED |
发明人 |
TANOURY GERALD J.;CHEN MINZHANG;JONES ANDREW D.;NYCE PHILIP L.;TRUDEAU MARTIN;GUERIN DAVID J.;SNOONIAN JOHN R. |
分类号 |
C07D405/12;A61K31/4025;C07B43/04;C07B57/00;C07D405/14 |
主分类号 |
C07D405/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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