发明名称 |
NEW POLYMORPHIC FORM OF IMATINIB BASE AND PREPARATION OF SALTS THEREOF |
摘要 |
The invention relates to a process for the manufacture of new polymorph of imatinib base, the preparation of mesylate salt thereof and their inclusion into pharmaceutical compositions which have an improved stability and purity, as well as processes for their preparation. |
申请公布号 |
WO2011157450(A1) |
申请公布日期 |
2011.12.22 |
申请号 |
WO2011EP03025 |
申请日期 |
2011.06.17 |
申请人 |
KRKA, D. D., NOVO MESTO;BENKIC PRIMOZ;TIHI JAROSLAV;PECAVAR ANICA;GERMAN TAMARA;VRECER FRANC;VAJS ANAMARIJA;SKRABANJA VIDA |
发明人 |
BENKIC PRIMOZ;TIHI JAROSLAV;PECAVAR ANICA;GERMAN TAMARA;VRECER FRANC;VAJS ANAMARIJA;SKRABANJA VIDA |
分类号 |
C07D401/04;A61K31/505;A61P35/00 |
主分类号 |
C07D401/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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