发明名称 PIPERIDINONE DERIVATIVES AS MDM2 INHIBITORS FOR THE TREATMENT OF CANCER
摘要 The present invention provides MDM2 inhibitor compounds of Formula (I), wherein the variables are defined above, which compounds are useful as therapeutic agents, particularly for the treatment of cancers. The present invention also relates to pharmaceutical compositions that contain an MDM2 inhibitor.
申请公布号 WO2011153509(A1) 申请公布日期 2011.12.08
申请号 WO2011US39184 申请日期 2011.06.03
申请人 AMGEN INC.;BARTBERGER, MICHAEL DAVID;GONZALEZ BUENROSTRO, ANA;BECK, HILARY PLAKE;CHEN, XIAOQI;CONNORS, RICHARD VICTOR;DEIGNAN, JEFFERY;DUQUETTE, JASON;EKSTEROWICZ, JOHN;FISHER, BENJAMIN;FOX, BRIAN MATTHEW;FU, JIASHENG;FU, ZICE;GONZALEZ LOPEZ DE TURISO, FELIX;GRIBBLE, JR., MICHAEL WILLIAM;GUSTIN, DARIN JAMES;HEATH, JULIE ANNE;HUANG, XIN;JIAO, XIANYUN;JOHNSON, MICHAEL;KAYSER, FRANK;KOPECKY, DAVID JOHN;LAI, SUJEN;LI, YIHONG;LI, ZHIHONG;LIU, JIWEN;LOW, JONATHAN DANTE;LUCAS, BRIAN STUART;MA, ZHIHUA;MCGEE, LAWRENCE;MCINTOSH, JOEL;MCMINN, DUSTIN;MEDINA, JULIO CESAR;MIHALIC, JEFFREY THOMAS;OLSON, STEVEN HOWARD;REW, YOSUP;ROVETO, PHILIP MARLEY;SUN, DAQING;WANG, XIAODONG;WANG, YINGCAI;YAN, XUELEI;YU, MING;ZHU, JIANG 发明人 BARTBERGER, MICHAEL DAVID;GONZALEZ BUENROSTRO, ANA;BECK, HILARY PLAKE;CHEN, XIAOQI;CONNORS, RICHARD VICTOR;DEIGNAN, JEFFERY;DUQUETTE, JASON;EKSTEROWICZ, JOHN;FISHER, BENJAMIN;FOX, BRIAN MATTHEW;FU, JIASHENG;FU, ZICE;GONZALEZ LOPEZ DE TURISO, FELIX;GRIBBLE, JR., MICHAEL WILLIAM;GUSTIN, DARIN JAMES;HEATH, JULIE ANNE;HUANG, XIN;JIAO, XIANYUN;JOHNSON, MICHAEL;KAYSER, FRANK;KOPECKY, DAVID JOHN;LAI, SUJEN;LI, YIHONG;LI, ZHIHONG;LIU, JIWEN;LOW, JONATHAN DANTE;LUCAS, BRIAN STUART;MA, ZHIHUA;MCGEE, LAWRENCE;MCINTOSH, JOEL;MCMINN, DUSTIN;MEDINA, JULIO CESAR;MIHALIC, JEFFREY THOMAS;OLSON, STEVEN HOWARD;REW, YOSUP;ROVETO, PHILIP MARLEY;SUN, DAQING;WANG, XIAODONG;WANG, YINGCAI;YAN, XUELEI;YU, MING;ZHU, JIANG
分类号 C07D211/40;A61K31/4412;A61P35/00;C07D279/02;C07D401/04;C07D401/06;C07D401/12;C07D407/04;C07D407/06;C07D409/04;C07D413/06;C07D417/06;C07D471/20;C07D498/08;C07D498/20 主分类号 C07D211/40
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