发明名称 SOLID FORMS OF [4-(3-FLUORO-5-TRIFLUOROMETHYL-PYRIDIN-2-YL)-PIPERAZIN-1-YL-[5-METHANESULFONYL-2-((S)-2,2,2-TRIFLUORO-1-METHYL-ETHOXY)-PHENYL]-METHANONE
摘要 The present invention relates to four distinct crystalline forms and to an amorphous form of [4-(3-Fluoro-5-trifluoromethyl-pyridin-2-yl)-piperazin-1-yl]-[5-methanesulfonyl-2-((S)-2,2,2-trifluoro-1-methyl-ethoxy)-phenyl]-methanone, and to their use in the preparation of pharmaceutical compositions. The compounds of present invention are suitable for the treatment of psychoses, pain, neurodegenerative disfunction in memory and learning, schizophrenia, dementia and other diseases in which cognitive processes are impaired, such as attention deficit disorders or Alzheimer's disease.
申请公布号 US2011295007(A1) 申请公布日期 2011.12.01
申请号 US201113188486 申请日期 2011.07.22
申请人 BUBENDORF ANDRE;DEYNET-VUCENOVIC ANNETTE;DIODONE RALPH;GRASSMANN OLAF;LINDENSTRUTH KAI;PINARD EMMANUEL;ROHRER FRANZISKA E.;SCHWITTER URS 发明人 BUBENDORF ANDRE;DEYNET-VUCENOVIC ANNETTE;DIODONE RALPH;GRASSMANN OLAF;LINDENSTRUTH KAI;PINARD EMMANUEL;ROHRER FRANZISKA E.;SCHWITTER URS
分类号 C07D401/04 主分类号 C07D401/04
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