发明名称 HETEROCYCLIC RING COMPOUND AND H1 RECEPTOR ANTAGONIST
摘要 Disclosed is a heterocyclic ring compound which is useful as an anti-allergic agent. Specifically disclosed is a compound represented by formula (1) or a salt thereof. (In the formula, the ring A represents an isocyclic or heterocyclic ring; the ring B represents a heterocyclic ring containing G and a nitrogen atom N as the ring-constituting atoms, wherein G in the ring B represents CH or N; R1 represents a carbonyl group or an alkylene group; R2a and R2b independently represent an alkyl group, a cycloalkyl group, an aryl group or a heterocyclic ring group; X represents an oxygen atom or a sulfur atom; Z represents a hydroxyl group, an alkoxy group, a cycloalkyloxy group, an aryloxy group, an aralkyloxy group, an amino group, or an N-substituted amino group; and n represents 0 or 1, wherein R1 represents an alkylene group which may have a substituent when the ring A represents a benzene ring or the ring B represents a piperazine ring.)
申请公布号 WO2011148888(A1) 申请公布日期 2011.12.01
申请号 WO2011JP61734 申请日期 2011.05.23
申请人 ASKA PHARMACEUTICAL CO., LTD.;OKADA MAKOTO;HASUMI KOICHI;NISHIMOTO TAKAHIRO;YOSHIDA MIWA;ISHITANI KOUKI;AOTSUKA TOMOJI;KANAZAWA HASHIME 发明人 OKADA MAKOTO;HASUMI KOICHI;NISHIMOTO TAKAHIRO;YOSHIDA MIWA;ISHITANI KOUKI;AOTSUKA TOMOJI;KANAZAWA HASHIME
分类号 C07D211/46;A61K31/4439;A61K31/445;A61K31/4525;A61K31/4535;A61K31/454;A61K31/4545;A61K31/455;A61K31/496;A61K31/497;A61P29/00;A61P37/08;A61P43/00;C07D213/79;C07D333/40;C07D401/06;C07D407/08;C07D409/06;C07D413/06;C07D417/06 主分类号 C07D211/46
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