发明名称 Fused heteroaryl derivatives
摘要 The present invention provides a pharmaceutical composition which is useful as a phosphatidylinositol 3 kinase (PI3K) inhibitor and an antitumor agent, and it provides a novel bicyclic or tricyclic fused heteroaryl derivative or a salt thereof which possesses an excellent PI3K inhibiting activity and cancer cell growth inhibiting activity.
申请公布号 US8067586(B2) 申请公布日期 2011.11.29
申请号 US20100688272 申请日期 2010.01.15
申请人 HAYAKAWA MASAHIKO;KAIZAWA HIROYUKI;MORITOMO HIROYUKI;KAWAGUCHI KEN-ICHI;KOIZUMI TOMONOBU;YAMANO MAYUMI;MATSUDA KOYO;OKADA MINORU;OHTA MITSUAKI;ASTELLAS PHARMA INC.;LUDWIG INSTITUTE FOR CANCER RESEARCH;IMPERIAL CANCER RESEARCH TECHNOLOGY LTD. 发明人 HAYAKAWA MASAHIKO;KAIZAWA HIROYUKI;MORITOMO HIROYUKI;KAWAGUCHI KEN-ICHI;KOIZUMI TOMONOBU;YAMANO MAYUMI;MATSUDA KOYO;OKADA MINORU;OHTA MITSUAKI
分类号 C07D413/00;A61K31/00;A61K31/517;A61K31/519;A61K31/5377;C07D471/04;C07D471/14;C07D491/04;C07D491/14;C07D495/04;C07D495/14 主分类号 C07D413/00
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