发明名称 PROCESS FOR THE PREPARATION OF CHIRAL TRIAZOLONES
摘要 A process for the preparation of a chiral compound, in particular posaconazole, wherein the process comprises mixing and reacting the compounds of formula (I) Y3-NH2; of formula (Ila) 0=C=N-Y0 and/or of formula (lIb) and of formula (III) in a solvent in any order to obtain a reaction mixture containing a chiral compound of formula (IV) and/or formula (V).
申请公布号 WO2011144653(A1) 申请公布日期 2011.11.24
申请号 WO2011EP58033 申请日期 2011.05.18
申请人 SANDOZ AG;OBERHUBER, MICHAEL;SALCHENEGGER, JOERG;DE SOUZA, DOMINIC;ALBERT, MARTIN;WILHELM, THORSTEN;LANGNER, MARTIN;STURM, HUBERT;SPITZENSTAETTER, HANS-PETER 发明人 OBERHUBER, MICHAEL;SALCHENEGGER, JOERG;DE SOUZA, DOMINIC;ALBERT, MARTIN;WILHELM, THORSTEN;LANGNER, MARTIN;STURM, HUBERT;SPITZENSTAETTER, HANS-PETER
分类号 C07D405/14;A61K31/496;A61P31/10 主分类号 C07D405/14
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