发明名称 |
VITAMIN E CONJUGATES, AND THEIR USES AS ANTIOXIDANTS AND PRODRUG DELIVERY VEHICLES |
摘要 |
<p>Tocopherol conjugates are disclosed that are useful as antioxidants or as pro-drug delivery vehicles. The conjugates are amphiphilic, and tend to localize at the interface between water domains and lipid domains. A prototype embodiment disclosed is an alpha tocopherol-linker-carnosine conjugate that has been designated VECAR.</p> |
申请公布号 |
CA2816928(A1) |
申请公布日期 |
2011.11.24 |
申请号 |
CA20112816928 |
申请日期 |
2011.05.18 |
申请人 |
BOARD OF SUPERVISORS OF LOUISIANA STATE UNIVERSITY AND AGRICULTURAL AND MECHANICAL COLLEGE |
发明人 |
SABLIOV, CRISTINA M.;ASTETE, CARLOS E.;SPIVAK, DAVID |
分类号 |
C07D405/12;A61K9/16;A61K31/4178;A61P9/00;A61P25/28;A61P35/00;C07D311/04 |
主分类号 |
C07D405/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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