发明名称 Nitrogenous heterocyclic compounds, preparation thereof and use thereof as antibacterial medicaments
摘要 The invention concerns nitrogenated heterocyclic compounds, their preparation and use as antibacterial drugs, compounds of general formula (I) wherein R1 represents a (CH2)n-NHR2 or (CH2)n-NHR radical, where R is a (C1-C6) alkyl and n is equal to 1 or 2; R2 represents a hydrogen atom; R3 and R4 together form an aromatic nitrogenated heterocycle with 5 apexes with 1, 2 or 3 nitrogen atoms optionally substituted by one or several R′ groups, R′ being selected in the group composed of a hydrogen atom and alkyl radicals with 1 to 6 carbon atoms; in free form, as zwitterions, and in the form of salts of pharmaceutically acceptable inorganic or organic bases and acids.
申请公布号 US8063219(B2) 申请公布日期 2011.11.22
申请号 US20080595120 申请日期 2008.04.11
申请人 LAMPILAS MAXIME;ROWLANDS DAVID ALUN;KEBSI ADEL;LEDOUSSAL BENOIT;PIERRES CAMILLE;NOVEXEL 发明人 LAMPILAS MAXIME;ROWLANDS DAVID ALUN;KEBSI ADEL;LEDOUSSAL BENOIT;PIERRES CAMILLE
分类号 A61K31/437;A61P31/04;C07D471/04 主分类号 A61K31/437
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