HETEROCYCLIC SULFONE MGLUR4 ALLOSTERIC POTENTIATORS, COMPOSITIONS, AND METHODS OF TREATING NEUROLOGICAL DYSFUNCTION
摘要
<p>Heterocyclic sulfone compounds which are useful as allosteric potentiators/positive allosteric modulators of the metabotropic glutamate receptor subtype 4 (mGluR4); and methods of using the compounds, for example, in treating neurological and psychiatric disorders or other disease state associated with glutamate dysfunction.</p>
申请公布号
CA2798514(A1)
申请公布日期
2011.11.17
申请号
CA20112798514
申请日期
2011.05.12
申请人
VANDERBILT UNIVERSITY
发明人
CONN, P. JEFFREY;LINDSLEY, CRAIG W.;HOPKINS, COREY R.;WEAVER, CHARLES DAVID;NISWENDER, COLLEEN M.;GOGLIOTTI, ROCCO D.;CHEUNG, YIU-YIN;SALOVICH, JAMES M.;ENGERS, DARREN W.